Aza-Wittig Reaction: Mechanism | Examples

The reaction of aza-ylides ( also called as iminophosphoranes) with different carbonyl molecules is called the
aza-Wittig reaction. In this post described the Aza-Wittig Reaction Mechanism with Examples.

Aza-Wittig Reaction
Aza-Wittig Reaction

Aza-Wittig Reaction Mechanism

Mechanism of Aza-Wittig Reaction are defined in two steps as follow

First step : the PPh3 reacts with an alkyl-azide and generate an iminophosphorane by loosing of nitrogen N2 (also called Staudinger reaction).

Second step: the nucleophilic nitrogen of the iminophosphorane attacks the carbonyl group and four-membered intermediate (oxazaphosphetane) generate, from oxazaphosphetane product Schiff base and the by-product triphenylphosphine oxide are released. this is the Aza-Wittig Reaction Mechanism

Aza-Wittig Reaction Mechanism
Aza-Wittig Reaction Mechanism

Aza-Wittig Reaction Examples:

Aza-Wittig Reaction with Mechanism and Examples has been shown below

Aza-Wittig Reaction Examples
Aza-Wittig Reaction Examples

Related Reactions:

  1. Wittig Reaction
  2. Staudinger Reaction

References:

  1. Catalytic Wittig and aza-Wittig reactions ^
  2. Strategic Applications of Named Reactions in Organic Synthesis ^^
  3. Aza-Wittig Reaction: Mechanism | Examples

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